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Opioid Receptor Three-Dimensional Structures from Distance Geometry Calculations with Hydrogen Bonding Constraints

Pogozheva, Irina D., Lomize, Andrei L., Mosberg, Henry I.

Journal:

Biophysical Journal

Année:

1998

Langue:

english

Fichier:

PDF, 759 KB

english, 1998

Complex of an Active μ-Opioid Receptor with a Cyclic Peptide Agonist Modeled from Experimental Constraints †

Fowler, Carol B., Pogozheva, Irina D., Lomize, Andrei L., LeVine, Harry, Mosberg, Henry I.

Journal:

Biochemistry

Année:

2004

Langue:

english

Fichier:

PDF, 627 KB

english, 2004

Further Optimization and Evaluation of Bioavailable, Mixed-Efficacy μ-Opioid Receptor (MOR) Agonists/δ-Opioid Receptor (DOR) Antagonists: Balancing MOR and DOR Affinities

Harland, Aubrie A., Yeomans, Larisa, Griggs, Nicholas W., Anand, Jessica P., Pogozheva, Irina D., Jutkiewicz, Emily M., Traynor, John R., Mosberg, Henry I.

Journal:

Journal of Medicinal Chemistry

Année:

2015

Langue:

english

Fichier:

PDF, 2.14 MB

english, 2015

In Vivo Effects of μ Opioid Receptor Agonist/δ Opioid Receptor Antagonist Peptidomimetics Following Acute and Repeated Administration

Anand, Jessica P, Kochan, Kelsey E, Nastase, Anthony F, Montgomery, Deanna, Griggs, Nicholas W, Traynor, John R, Mosberg, Henry I, Jutkiewicz, Emily M

Journal:

British Journal of Pharmacology

Année:

2018

Langue:

english

Fichier:

PDF, 1.16 MB

english, 2018

Prediction of protein structure: The problem of fold multiplicity

Andrei L. Lomize, Irina D. Pogozheva, Henry I. Mosberg

Journal:

Proteins: Structure, Function, and Bioinformatics

Année:

1999

Langue:

english

Fichier:

PDF, 154 KB

english, 1999

Development of a model for the δ-opioid receptor pharmacophore: 3. Comparison of the cyclic tetrapeptide Tyr-c[D-Cys-Phe-D-Pen] OH with other conformationally constrained δ-receptor selective ligands

Andrei L. Lomize, Irina D. Pogozheva, Henry I. Mosberg

Journal:

Biopolymers

Année:

1996

Langue:

english

Fichier:

PDF, 1.03 MB

english, 1996

Development of a model for the δ-opioid receptor pharmacophore. 4. Residue 3 dehydrophenylalanine analogues of Tyr-c[D-Cys-Phe-D-Pen]OH (JOM-13) confirm required gauche orientation of aromatic side chain

Henry I. Mosberg, Rajesh K. Dua, Irina D. Pogozheva, Andrei L. Lomize

Journal:

Biopolymers

Année:

1996

Langue:

english

Fichier:

PDF, 758 KB

english, 1996

Thermodynamic model of secondary structure for α-helical peptides and proteins

Andrei L. Lomize, Henry I. Mosberg

Journal:

Biopolymers

Année:

1997

Langue:

english

Fichier:

PDF, 272 KB

english, 1997

Complementarity of δ opioid ligand pharmacophore and receptor models

Henry I. Mosberg

Journal:

Biopolymers

Année:

1999

Langue:

english

Fichier:

PDF, 426 KB

english, 1999

Long-range spin–spin coupling as an aid for the assignment of aromatic residues in peptide 1H-nmr spectra

Henry I. Mosberg

Journal:

Biopolymers

Année:

1982

Langue:

english

Fichier:

PDF, 209 KB

english, 1982

Conformational and dynamic considerations in the design of peptide hormone analogs

Victor J. Hruby, Henry I. Mosberg, Tomi K. Sawyer, James J. Knittel, Todd W. Rockway, James Ormberg, Paul Darman, W. Y. Chan, Mac E. Hadley

Journal:

Biopolymers

Année:

1983

Langue:

english

Fichier:

PDF, 812 KB

english, 1983

Synthesis of deuterium labelled penicillamine and its use for the assignment of the 1H NMR spectra of two cyclic enkephalin analogs

Henry I. Mosberg, John R. Omnaas, Kondareddiar Ramalingam, Ronald W. Woodard

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Année:

1987

Langue:

english

Fichier:

PDF, 325 KB

english, 1987

Utilization of peptide carrier system to improve intestinal absorption: Targeting prolidase as a prodrug-converting enzyme

Jane P.-F. Bai, Ming Hu, P. Subramanian, Henry I. Mosberg, Gordon L. Amidon

Journal:

Journal of Pharmaceutical Sciences

Année:

1992

Langue:

english

Fichier:

PDF, 410 KB

english, 1992

Specifically deuterated l-malate as an NMR probe of the aspartate transcarbamylase catalytic site

Henry I Mosberg, Paul G Schmidt, Sally S Seaver

Journal:

Journal of Magnetic Resonance (1969)

Année:

1969

Langue:

english

Fichier:

PDF, 428 KB

english, 1969

Synthesis of a novel series of topographically constrained amino acids: Benzo-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids

Chenguang Wang, Henry I. Mosberg

Journal:

Tetrahedron Letters

Année:

1995

Langue:

english

Fichier:

PDF, 149 KB

english, 1995

1H NMR of succinate binding to aspartate transcarbamylase a comparison of results in D2O and H2O

Henry I. Mosberg, Carol B. Beard, Paul G. Schmidt

Journal:

Biophysical Chemistry

Année:

1976

Langue:

english

Fichier:

PDF, 849 KB

english, 1976

A high affinity, mu-opioid receptor-selective enkephalin analogue lacking an N-terminal tyrosine

Henry I. Mosberg, Jeffrey C. Ho, Katarzyna Sobczyk-Kojiro

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1998

Langue:

english

Fichier:

PDF, 207 KB

english, 1998

Design of a high affinity peptidomimetic opioid agonist from peptide pharmacophore models

Chenguang Wang, Iain J. McFadyen, John R. Traynor, Henry I. Mosberg

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1998

Langue:

english

Fichier:

PDF, 205 KB

english, 1998

Key Residues Defining the μ-Opioid Receptor Binding Pocket: A Site-Directed Mutagenesis Study

Alfred Mansour, Larry P. Taylor, Jeffrey L. Fine, Robert C. Thompson, Mary T. Hoversten, Henry I. Mosberg, Stanley J. Watson, Huda Akil

Journal:

Journal of Neurochemistry

Année:

1997

Langue:

english

Fichier:

PDF, 1.07 MB

english, 1997

A covalent peptide inhibitor of RGS4 identified in a focused one-bead, one compound library screen

Rebecca A Roof, David L Roman, Samuel T Clements, Katarzyna Sobczyk-Kojiro, Levi L Blazer, Shodai Ota, Henry I Mosberg, Richard R Neubig

Journal:

BMC Pharmacology

Année:

2009

Langue:

english

Fichier:

PDF, 1.20 MB

english, 2009

The role of hydrophobic interactions in positioning of peripheral proteins in membranes

Andrei L Lomize, Irina D Pogozheva, Mikhail A Lomize, Henry I Mosberg

Journal:

BMC Structural Biology

Année:

2007

Langue:

english

Fichier:

PDF, 6.72 MB

english, 2007

Pharmacophore elements of the TIPP class of delta opioid receptor antagonists

Henry I. Mosberg, John R. Omnaas, Katarzyna Sobczyk-Kojiro, Raj Dua, Jeffrey C. Ho, Wenli Ma, Paula Bush, Carol Mousigian, Andrei Lomize

Journal:

International Journal of Peptide Research and Therapeutics

Année:

1994

Langue:

english

Fichier:

PDF, 291 KB

english, 1994

Synthesis of 6- or 7-substituted 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids

Wenli Ma, Henry I. Mosberg

Journal:

International Journal of Peptide Research and Therapeutics

Année:

1999

Langue:

english

Fichier:

PDF, 390 KB

english, 1999

Molecular Mechanism of the Constitutive Activation of the L250Q Human Melanocortin-4 Receptor Polymorphism

Bettina Proneth, Zhimin Xiang, Irina D. Pogozheva, Sally A. Litherland, Oleg S. Gorbatyuk, Amanda M. Shaw, William J. Millard, Henry I. Mosberg, Carrie Haskell-Luevano

Journal:

Chemical Biology & Drug Design

Année:

2006

Langue:

english

Fichier:

PDF, 959 KB

english, 2006

Mechanism of Action and Structural Requirements of Constrained Peptide Inhibitors of RGS Proteins

Rebecca A. Roof, Yafei Jin, David L. Roman, Roger K. Sunahara, Masaru Ishii, Henry I. Mosberg, Richard R. Neubig

Journal:

Chemical Biology & Drug Design

Année:

2006

Langue:

english

Fichier:

PDF, 365 KB

english, 2006

Synthesis of Novel Peptide Inhibitors of Thrombin-induced Platelet Activation

Fernanda M. Burke, Mark Warnock, Alvin H. Schmaier, Henry I. Mosberg

Journal:

Chemical Biology & Drug Design

Année:

2006

Langue:

english

Fichier:

PDF, 63 KB

english, 2006

Novel Peptide Ligands of RGS4 from a Focused One-Bead, One-Compound Library

Rebecca A. Roof, Katarzyna Sobczyk-Kojiro, Anjanette J. Turbiak, David L. Roman, Irina D. Pogozheva, Levi L. Blazer, Richard R. Neubig, Henry I. Mosberg

Journal:

Chemical Biology & Drug Design

Année:

2008

Langue:

english

Fichier:

PDF, 369 KB

english, 2008

Structure-Based Design of Residue 1 Analogs of the Direct Thrombin Inhibitor Pentapeptide FM 19

Elizabeth A. Girnys, Katarzyna Sobczyk-Kojiro, Henry I. Mosberg

Journal:

Chemical Biology & Drug Design

Année:

2010

Langue:

english

Fichier:

PDF, 167 KB

english, 2010

Structural organization of G-protein-coupled receptors

Andrei L. Lomize, Irina D. Pogozheva, Henry I. Mosberg

Journal:

Journal of Computer-Aided Molecular Design

Année:

1999

Langue:

english

Fichier:

PDF, 659 KB

english, 1999

Synthesis of 6- or 7-substituted 1,2,3,4-tetrahydroisoquinoline- 3-carboxylic acids

Wenli Ma, Henry I. Mosberg

Journal:

International Journal of Peptide Research and Therapeutics

Année:

1999

Langue:

english

Fichier:

PDF, 49 KB

Ming Hu, Pullachipatti Subramanian, Henry I. Mosberg, Gordon L. Amidon

Journal:

Pharmaceutical Research

Année:

1989

Fichier:

PDF, 776 KB

1989

SYNTHESIS, PHARMACOLOGICAL, CONFORMATIONAL, AND DYNAMIC STUDIES OF THE POTENT HORMONE ANTAGONISTS [1-PENICILLAMINE, 4-THREONINE]-OXYTOCIN AND [1-PENICILLAMINE, 2-PHENYLALANINE, 4-THREONINE] -OXYTOCIN : Conformational and Dynamic Considerations in the Design of Antagonists

VICTOR J. HRUBY, HENRY I. MOSBERG, MAC E. HADLEY, W. Y. CHAN, ANDREA M. POWELL

Journal:

Chemical Biology & Drug Design

Année:

1980

Langue:

english

Fichier:

PDF, 647 KB

english, 1980

1H n.m.r. investigation of conformational features of cyclic enkephalinamide analogs

Henry I. Mosberg, Peter W. Schiller

Journal:

Chemical Biology & Drug Design

Année:

1984

Langue:

english

Fichier:

PDF, 326 KB

english, 1984

1H-n.m.r. investigation of conformational features of cyclic, penicillamine-containing enkephalin analogs

HENRY I. MOSBERG

Journal:

Chemical Biology & Drug Design

Année:

1987

Langue:

english

Fichier:

PDF, 478 KB

english, 1987

Role of steric interactions in the delta opioid receptor selectivity of [d-Pen2, d-Pen5]enkephalin

HENRY I. MOSBERG, RONALD C. HAASETH, KONDAREDDIAR RAMALINGAM, ALFRED MANSOUR, HUDA AKIL, RONALD W. WOODARD

Journal:

Chemical Biology & Drug Design

Année:

1988

Langue:

english

Fichier:

PDF, 525 KB

english, 1988

Single residue modifications of the delta opioid receptor selective peptide, [d-Pen2,d-Pen5]-enkephalin (DPDPE) : Correlation of pharmacological effects with structural and conformational features

RONALD C. HAASETH, KATARZYNA SOBCZYK-KOJIRO, FEDOR MEDZIHRADSKY, CHARLES B. SMITH, HENRY I. MOSBERG

Journal:

Chemical Biology & Drug Design

Année:

1990

Langue:

english

Fichier:

PDF, 703 KB

english, 1990

Opioid receptor affinity and selectivity effects of second residue and carboxy terminal residue variation in a cyclic disulfide-containing opioid tetrapeptide

DEBORAH L. HEYL, JOHN R. OMNAAS, KATARZYNA SOBCZYK-KOJIRO, FEDOR MEDZIHRADSKY, CHARLES B. SMITH, HENRY I. MOSBERG

Journal:

Chemical Biology & Drug Design

Année:

1991

Langue:

english

Fichier:

PDF, 592 KB

english, 1991

Modification of the Phe3 aromatic moiety in delta receptor-selective dermorphin/deltorphin-related tetrapeptides Effects on opioid receptor binding

DEBORAH L. HEYL, HENRY I. MOSBERG

Journal:

Chemical Biology & Drug Design

Année:

1992

Langue:

english

Fichier:

PDF, 796 KB

english, 1992

Raman study of crystalline peptides containing β turns

Jay A. Fox, Anthony T. Tu, Victor J. Hruby, Henry I. Mosberg

Journal:

Archives of Biochemistry and Biophysics

Année:

1981

Langue:

english

Fichier:

PDF, 349 KB

english, 1981

[D-Pen2, L-cys5]enkephalinamide and [D-pen2, D-cys5]enkephalinamide, conformationally constrained cyclic enkephalinamide analogs with delta receptor specificity

Henry I. Mosberg, Robin Hurst, Victor J. Hruby, James J. Galligan, Thomas F. Burks, Kelvin Gee, Henry I. Yamamura

Journal:

Biochemical and Biophysical Research Communications

Année:

1982

Langue:

english

Fichier:

PDF, 449 KB

english, 1982

Opioid δ-receptor involvement in supraspinal and spinal antinociception in mice

Julius S. Heyman, Sheila A. Mulvaney, Henry I. Mosberg, Frank Porreca

Journal:

Brain Research

Année:

1987

Langue:

english

Fichier:

PDF, 684 KB

english, 1987

Modulation of μ-mediated antinociception by δ agonists in the mouse: selective potentiation of morphine and normorphine by [D-Pen2, D-Pen5]enkephalin

Julius S. Heyman, Jeffry L. Vaught, Henry I. Mosberg, Ronald C. Haaseth, Frank Porreca

Journal:

European Journal of Pharmacology

Année:

1989

Langue:

english

Fichier:

PDF, 733 KB

english, 1989